SCHEMBL8638460

SCHEMBL8638460

COc1cc(C(=O)Nc2ccccc2C(N)=O)cc(OC)c1OC

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.65
LMNA P02545 4/20 0.65
CHEK1 O14757 1/20 0.62
PIM1 P11309 1/20 0.62
MAPK8 P45983 1/20 0.62
CLK4 Q9HAZ1 1/20 0.62
ABCB1 P08183 3/20 0.59
ALDH1A1 P00352 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
HPGD P15428 2/20 0.57
HTT P42858 1/20 0.57
KDM4E B2RXH2 1/20 0.55
HSD17B10 Q99714 1/20 0.55
PKM P14618 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367182 0.88 CHEK1 (0.80) LMNACHEK1PIM1MAPK8CLK4
SCHEMBL4699872 0.88 CHEK1 (0.76) L3MBTL1LMNACHEK1PIM1MAPK8
SCHEMBL8635556 0.83 KDM4E (0.77) CHEK1PIM1MAPK8CLK4ALDH1A1
SCHEMBL8638027 0.82 MEN1 (0.67) LMNAALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL22340657 0.81 TSHR (0.75) LMNASMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL4523815 0.81 MAPK9 (0.76) LMNACHEK1PIM1MAPK8CLK4
SCHEMBL24489009 0.81 KMT2A (0.80) LMNACHEK1PIM1MAPK8CLK4
SCHEMBL29579206 0.81 KMT2A (0.80) LMNACHEK1PIM1MAPK8CLK4
SCHEMBL14256345 0.80 L3MBTL1 (0.58) L3MBTL1LMNACHEK1PIM1MAPK8
SCHEMBL8641094 0.80 KMT2A (0.57) LMNAALDH1A1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4225745-A1 ACETAMIDO-PHENYLBENZAMIDE DERIVATIVES AND METHODS OF USING THE SAME Athenex, Inc. (US) 2023-08-16 EP disclosed
WO-2022076662-A1 ACETAMIDO-PHENYLBENZAMIDE DERIVATIVES AND METHODS OF USING THE SAME ATHENEX, INC. (US) 2022-04-14 WO disclosed
EP-0855387-A1 2-ACYLAMINOBENZAMIDE DERIVATIVES AND PREVENTIVE AND REMEDY FOR DISEASES CAUSED BY THE SUPERMULTIPLICATION OF VASCULAR INTIMAL CELLS KISSEI PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed