SCHEMBL8638646

SCHEMBL8638646

CCCCCc1cc(F)c(B2OCC(CCCC)CO2)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.38
CYP3A4 P08684 1/20 0.38
SPHK2 Q9NRA0 7/20 0.32
SPHK1 Q9NYA1 5/20 0.32
LPL P06858 5/20 0.32
LIPG Q9Y5X9 5/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
GPR84 Q9NQS5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8642283 0.97 PTGS2 (0.35) PTGS2CYP3A4SPHK2SPHK1LPL
SCHEMBL8636432 0.96 PTGS2 (0.36) PTGS2CYP3A4SPHK2SPHK1LPL
SCHEMBL8637758 0.96 PTGS2 (0.36) PTGS2CYP3A4SPHK2SPHK1LPL
SCHEMBL8639954 0.95 PTGS2 (0.35) PTGS2CYP3A4SPHK2SPHK1LPL
SCHEMBL8642880 0.93
SCHEMBL8645125 0.92 CYP1A2 (0.31)
SCHEMBL8641996 0.91 ALDH1A1 (0.33) PTGS2
SCHEMBL8642971 0.91 ALDH1A1 (0.33) PTGS2
SCHEMBL8640268 0.90 PTGS2 (0.36) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8642159 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440082-B1 Method for the conversion of fluorinated aromatic compounds using electrophiles MERCK PATENT GMBH (DE) 1998-04-15 EP disclosed
US-5262556-A Alkylation or hydroxyalkylation by deprotonation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-11-16 US disclosed
EP-0440082-A2 Method for the conversion of fluorinated aromatic compounds using electrophiles MERCK PATENT GmbH (DE) 1991-08-07 EP disclosed