SCHEMBL8640268

SCHEMBL8640268

CCCCCc1cc(F)c(B2OCC(CC)CO2)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.36
CYP3A4 P08684 2/20 0.36
LPL P06858 5/20 0.33
LIPG Q9Y5X9 5/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
GPR84 Q9NQS5 2/20 0.33
ESR1 P03372 2/20 0.32
ADRA2A P08913 2/20 0.32
ADORA3 P0DMS8 2/20 0.32
TACR2 P21452 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
SHBG P04278 1/20 0.32
TP53 P04637 1/20 0.32
HSPD1 P10809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8638646 0.90 PTGS2 (0.38) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8639954 0.90 PTGS2 (0.35) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8642283 0.90 PTGS2 (0.35) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8640917 0.90 PKM (0.30)
SCHEMBL8636432 0.89 PTGS2 (0.36) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8637758 0.89 PTGS2 (0.36) PTGS2CYP3A4LPLLIPGTHRA
SCHEMBL8642971 0.84 ALDH1A1 (0.33) PTGS2ALDH1A1
SCHEMBL8641996 0.84 ALDH1A1 (0.33) PTGS2ALDH1A1
SCHEMBL8642880 0.83
SCHEMBL9571159 0.83 PTGS2 (0.36) PTGS2CYP3A4LPLLIPGTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440082-B1 Method for the conversion of fluorinated aromatic compounds using electrophiles MERCK PATENT GMBH (DE) 1998-04-15 EP disclosed
US-5262556-A Alkylation or hydroxyalkylation by deprotonation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-11-16 US disclosed
EP-0440082-A2 Method for the conversion of fluorinated aromatic compounds using electrophiles MERCK PATENT GmbH (DE) 1991-08-07 EP disclosed