SCHEMBL8639101

SCHEMBL8639101

CSc1ccc(-c2cc(C(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.52
PTGS1 P23219 10/20 0.52
ABCB11 O95342 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525009 0.88 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8637047 0.88 PTGS2 (0.63) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7928751 0.87 PTGS2 (0.66) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8165901 0.86 PTGS2 (0.62) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8635925 0.86 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7773921 0.85 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8625458 0.85 PTGS2 (0.67) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8688704 0.83 PTGS2 (0.51) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639180 0.83 PTGS2 (0.53) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7055102 0.83 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed