SCHEMBL8639776

SCHEMBL8639776

N#Cc1cc(-c2ccc([N+](=O)[O-])cc2)n(-c2ccccc2S(N)(=O)=O)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.49
CA12 O43570 5/20 0.48
CA9 Q16790 9/20 0.42
IKBKB O14920 1/20 0.40
CA2 P00918 7/20 0.39
CA1 P00915 5/20 0.39
CA14 Q9ULX7 2/20 0.39
CA13 Q8N1Q1 2/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PTGS1 P23219 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691511 0.86 PTGS2 (0.51) PTGS2CA12CA9CA2CA1
SCHEMBL8693252 0.84 PTGS2 (0.65) PTGS2CA12CA9CA2CA1
SCHEMBL8637414 0.84 PTGS2 (0.50) PTGS2CA12CA9CA2CA1
SCHEMBL8421758 0.84 PTGS2 (0.49) PTGS2CA12CA9CA2CA1
SCHEMBL8640732 0.84 PTGS2 (0.50) PTGS2CA2PTGS1CA7PDPK1
SCHEMBL8689658 0.84 PTGS2 (0.50) PTGS2CA12CA9CA2CA1
SCHEMBL8689144 0.83 PTGS2 (0.48) PTGS2CA9CA2CA1PTGS1
SCHEMBL8640581 0.82 PTGS2 (0.69) PTGS2CA12CA9CA2CA1
SCHEMBL6343738 0.81 PTGS2 (0.73) PTGS2CA12CA9CA2CA1
SCHEMBL8422297 0.80 PTGS2 (0.50) PTGS2CA12CA9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed