SCHEMBL8689658

SCHEMBL8689658

Cc1ccc(-c2cc(C#N)nn2-c2ccccc2S(N)(=O)=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.50
CYP2C9 P11712 2/20 0.45
CA9 Q16790 5/20 0.41
CA2 P00918 4/20 0.41
CA1 P00915 3/20 0.41
CA12 O43570 3/20 0.41
PDPK1 O15530 2/20 0.41
PTGS1 P23219 2/20 0.41
PTGES O14684 1/20 0.41
HDAC3 O15379 1/20 0.41
PDE5A O76074 1/20 0.41
ABCB11 O95342 1/20 0.41
MT-CO2 P00403 1/20 0.41
LMNA P02545 1/20 0.41
CA3 P07451 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX5 P09917 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691511 0.90 PTGS2 (0.51) PTGS2CYP2C9CA9CA2CA1
SCHEMBL8689144 0.89 PTGS2 (0.48) PTGS2CA9CA2CA1PTGS1
SCHEMBL8640732 0.88 PTGS2 (0.50) PTGS2CA2PDPK1PTGS1CA7
SCHEMBL8693252 0.88 PTGS2 (0.65) PTGS2CA9CA2CA1CA12
SCHEMBL8637414 0.88 PTGS2 (0.50) PTGS2CA9CA2CA1CA12
SCHEMBL8639776 0.84 PTGS2 (0.49) PTGS2CA9CA2CA1CA12
Benzenesulfonamide SCHEMBL7929456 0.84 PTGS2 (0.68) PTGS2CA9CA2CA1PDPK1
SCHEMBL8420750 0.83 CYP2C9 (0.63) PTGS2CYP2C9CA9CA2CA1
SCHEMBL8689204 0.82 PTGS2 (0.38) PTGS2CA9CA2CA1CA12
SCHEMBL8689101 0.82 PTGS2 (0.42) PTGS2CA9CA2CA1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed