SCHEMBL8640683

SCHEMBL8640683

COc1ccc(CS)c(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.48
APLNR P35414 1/20 0.44
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ADRA1A P35348 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2A6 P11509 1/20 0.39
POLB P06746 1/20 0.39
ESR1 P03372 1/20 0.38
CYP19A1 P11511 1/20 0.38
ESR2 Q92731 1/20 0.38
CRHR1 P34998 1/20 0.37
HDAC3 O15379 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3484107 0.81 APLNR (0.46) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL30486651 0.81 APLNR (0.46) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL3527192 0.81 APLNR (0.46) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL6603605 0.79 APLNR (0.44) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL20446477 0.79 HTR2B (0.50) IDO1APLNRHTR2AHTR2CADRA1A
Ammonia Solution, Strong SCHEMBL10346000 0.79 APLNR (0.44) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL3258877 0.79 IDO1 (0.48) IDO1APLNRCA12CA1CA2
SCHEMBL3963106 0.79 APLNR (0.63) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL6804542 0.79 ALDH1A1 (0.49) IDO1APLNRHTR2AHTR2CCA12
SCHEMBL9171486 0.79 APLNR (0.44) IDO1APLNRHTR2AHTR2CCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0516257-B1 Phenylbenzo[b]furans and -thiophenes, procedures for their preparation, and pharmaceutical compositions containing the same SCHERING AG (DE) 1998-08-05 EP disclosed
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
WO-1992021669-A1 2-PHENYLBENZO[B]FURANS AND THIOPHENES, METHODS OF PREPARING THEM AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM SCHERING AKTIENGESELLSCHAFT (DE) 1992-12-10 WO disclosed
EP-0516257-A1 Phenylbenzo[b]furans and -thiophenes, procedures for their preparation, and pharmaceutical compositions containing the same SCHERING AKTIENGESELLSCHAFT (DE) 1992-12-02 EP disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed