SCHEMBL8640754

SCHEMBL8640754

COc1cc(C(=O)N2CCC(c3ccc(F)c(F)c3)C2)cc(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.53
GAA P10253 1/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 1/20 0.50
UBE2M P61081 1/20 0.49
DCUN1D1 Q96GG9 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PDE2A O00408 1/20 0.48
POLB P06746 1/20 0.48
ROCK2 O75116 1/20 0.47
HTT P42858 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8352641 0.87 PDE4B (0.65) PDE4BGAA
SCHEMBL8638316 0.86 SCD5 (0.55) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8636998 0.85 ALDH1A1 (0.65) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8347627 0.84 PDE4B (0.53) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8640542 0.84 PDE4B (0.56) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8351152 0.84 ALDH1A1 (0.64) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8638632 0.83 PDE4B (0.53) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8635894 0.83 PROKR1 (0.53) PDE4BGAAALDH1A1CYP1A2UBE2M
SCHEMBL8351389 0.82 ALDH1A1 (0.56) GAAALDH1A1CYP1A2UBE2MDCUN1D1
SCHEMBL8355588 0.81 KMT2A (0.54) PDE4BGAAALDH1A1CYP1A2UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed