SCHEMBL8640795

SCHEMBL8640795

CSc1ccc(-c2cc(N)nn2-c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.50
KDM5B Q9UGL1 1/20 0.50
PTGS2 P35354 4/20 0.48
PTGS1 P23219 1/20 0.48
RPA1 P27694 4/20 0.47
RARG P13631 4/20 0.47
RXRA P19793 4/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
PPP1CA P62136 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
RECQL P46063 1/20 0.42
RARA P10276 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641532 0.82 PTGS2 (0.69) PTGS2PTGS1MAPTCYP2C9
SCHEMBL7456119 0.82 PTGS2 (0.67) PTGS2PTGS1RPA1RARGRXRA
SCHEMBL8645116 0.82 MALT1 (0.50) PTGS2PTGS1RPA1ALDH1A1SMN1; SMN2
SCHEMBL9202494 0.82 PTGS2 (0.52) PTGS2PTGS1SMN1; SMN2NPC1RAB9A
SCHEMBL7465856 0.80 PTGS2 (0.54) PTGS2PTGS1RPA1CYP1A2CYP2C9
SCHEMBL7872838 0.80 PTGS2 (0.47) PTGS2PTGS1RPA1ALDH1A1SMN1; SMN2
SCHEMBL7867785 0.80 PTGS2 (0.47) PTGS2PTGS1SMN1; SMN2NPC1RAB9A
SCHEMBL8639378 0.79 PTGS2 (0.53) PTGS2PTGS1ALDH1A1HPGDSMN1; SMN2
SCHEMBL8923289 0.78 CA9 (0.58) RPA1ALDH1A1HPGDSMN1; SMN2TP53
SCHEMBL7874456 0.78 PTGS2 (0.46) PTGS2PTGS1ALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0856000-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-05 EP disclosed
WO-1997013755-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-17 WO disclosed