SCHEMBL8641971

SCHEMBL8641971

CCOC(=O)c1nn(C)c(OC(F)F)c1C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
USP2 O75604 1/20 0.37
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
PDE4D Q08499 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
ELANE P08246 2/20 0.35
MEN1 O00255 2/20 0.35
GAA P10253 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL537675 0.86 ALDH1A1 (0.35) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL8652790 0.81 KDM4E (0.33) KDM4E
SCHEMBL8623813 0.80 GRM5 (0.31)
SCHEMBL1412582 0.79 TP53 (0.42) KMT2ARAB9AKDM4ESMN1; SMN2MEN1
SCHEMBL22900489 0.76 KMT2A (0.46) KMT2AUSP2NPC1RAB9AALDH1A1
SCHEMBL12682954 0.75 ADORA1 (0.42) KMT2AUSP2NPC1RAB9AALDH1A1
SCHEMBL1412587 0.75 ELANE (0.39) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL3797706 0.74 ADORA3 (0.41) KMT2AUSP2NPC1RAB9AALDH1A1
SCHEMBL12683029 0.74 CYP1A2 (0.46) KMT2AUSP2NPC1RAB9AALDH1A1
SCHEMBL4700865 0.73 ADORA3 (0.47) KMT2ANPC1RAB9AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923558-A1 SUBSTITUTED 1-(3-PYRAZOLYL)-PYRAZOLES BAYER AG (DE) 1999-06-23 EP disclosed
WO-1998006702-A1 SUBSTITUTED 1-(3-PYRAZOLYL)-PYRAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1998-02-19 WO disclosed