SCHEMBL8642030

SCHEMBL8642030

OC(c1ccc(F)cc1)[C@H]1CC[C@H]2CN(CC3CC3)CCN2C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.45
HTR2C P28335 2/20 0.45
HTR7 P34969 2/20 0.45
CYP2D6 P10635 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
HTR6 P50406 1/20 0.40
SLC6A2 P23975 1/20 0.39
KCNH2 Q12809 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641073 0.81 HTR2A (0.58) HTR2AHTR2CHTR7CYP2D6HTR6
SCHEMBL467404 0.75 KDM2B (0.53) HTR2AHTR2CHTR7HTR6DRD2
SCHEMBL8646880 0.75 KDM2B (0.53) HTR2AHTR2CHTR7HTR6DRD2
SCHEMBL467405 0.75 KDM2B (0.53) HTR2AHTR2CHTR7HTR6DRD2
SCHEMBL467403 0.75 KDM2B (0.53) HTR2AHTR2CHTR7HTR6DRD2
SCHEMBL14532757 0.74 DRD4 (0.57) HTR2ASLC6A2DRD2DRD4
SCHEMBL14502917 0.74 DRD4 (0.57) HTR2ASLC6A2DRD2DRD4
SCHEMBL5414076 0.74 DRD4 (0.57) HTR2ASLC6A2DRD2DRD4
SCHEMBL8642032 0.70 KDM4E (0.55)
SCHEMBL1348883 0.69 HTR2A (0.58) HTR2AHTR2CHTR7CYP2D6HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731307-A Neuroleptic 2,7-disubtituted perhydro-1h-pyrido 1, 2-A!pyrazines PFIZER, INC. (US) 1998-03-24 US claimed