SCHEMBL8645946

SCHEMBL8645946

O=C(NC(CSc1ccc2ccccc2c1)C(O)CCl)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
CASP1 P29466 3/20 0.44
CYP3A4 P08684 3/20 0.42
CYP2C19 P33261 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CTRB1 P17538 2/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
TOP2A P11388 1/20 0.40
TOP2B Q02880 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282041 1.00 CTSL (0.45) CTSLCTSBCTSSCASP1CYP3A4
SCHEMBL6629350 1.00 CTSL (0.45) CTSLCTSBCTSSCASP1CYP3A4
SCHEMBL7594853 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL5329730 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL6328905 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL6577081 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL7491284 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL6577088 0.89 CASP1 (0.48) CTSLCTSBCTSSCASP1CTRB1
SCHEMBL5230909 0.82 CASP1 (0.52) CTSLCTSBCTSSCASP1CYP3A4
SCHEMBL5226937 0.81 PPARA (0.55) CTSLCTSBCTSSCASP1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827891-A FOR TREATMENT OF AIDS, BLOCKING REPLICATION OF HIV VIRUS AGOURON PHARMACEUTICALS, INC. 1998-10-27 US disclosed