SCHEMBL8649236

SCHEMBL8649236

O=CCCc1ccc(Br)o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
TSHR P16473 2/20 0.35
POLB P06746 6/20 0.34
HPGD P15428 3/20 0.33
MAPT P10636 2/20 0.33
PKM P14618 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
GFER P55789 1/20 0.33
RECQL P46063 1/20 0.33
MCL1 Q07820 1/20 0.33
KMT2A Q03164 3/20 0.31
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 2/20 0.31
NSD2 O96028 1/20 0.31
DNMT1 P26358 1/20 0.31
APEX1 P27695 1/20 0.31
PPARG P37231 1/20 0.31
NCOA2 Q15596 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1616548 0.84 ALDH1A1 (0.41) ALDH1A1TSHRPOLBMAPTPKM
SCHEMBL1647691 0.78
SCHEMBL4155788 0.75 CHRM2 (0.45) ALDH1A1TSHRPOLBHPGDMAPT
SCHEMBL13680858 0.75 ALDH1A1 (0.35) ALDH1A1TSHRPOLBHPGDMAPT
SCHEMBL13680861 0.75 ALDH1A1 (0.35) ALDH1A1TSHR
SCHEMBL27876267 0.73
SCHEMBL25183771 0.71 HIF1A (0.41) ALDH1A1TSHR
SCHEMBL13543542 0.71
SCHEMBL8645128 0.71 ALDH1A1 (0.32) ALDH1A1TSHR
SCHEMBL25180381 0.70 EPHX2 (0.46) ALDH1A1TSHRHPGDMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-5808101-A 1,3-benzodioxole and 1,2-dialkoxybenzene derivatives as ocular hypotensive agents ALLERGAN (US) 1998-09-15 US disclosed
US-5710288-A 1,3-benzodioxole and 1,2-dialkoxybenzene derivatives as ocular hypotensive agents ALLERGAN (US) 1998-01-20 US disclosed