SCHEMBL8649367

SCHEMBL8649367

CCOC(=O)COc1cccc(C=C(C(=O)O)c2cccnc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.50
MEN1 O00255 4/20 0.50
ALDH1A1 P00352 3/20 0.50
LMNA P02545 1/20 0.47
THRB P10828 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GRM2 Q14416 1/20 0.46
MAPT P10636 3/20 0.45
HPGD P15428 2/20 0.45
CYP1A1 P04798 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP1B1 Q16678 1/20 0.45
TBXAS1 P24557 1/20 0.44
TSHR P16473 1/20 0.44
POLB P06746 1/20 0.44
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
KDM4E B2RXH2 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8649361 1.00 KMT2A (0.50) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL27520778 0.85 RAB9A (0.42) KMT2AMEN1ALDH1A1LMNATHRB
Hydrochloric Acid SCHEMBL8667384 0.84 RAB9A (0.41) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL8645503 0.82 ALDH1A1 (0.74) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8645501 0.82 ALDH1A1 (0.74) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8650792 0.82 ALDH1A1 (0.69) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL8650796 0.82 ALDH1A1 (0.69) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL8644315 0.80 KMT2A (0.56) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL8644310 0.80 KMT2A (0.56) KMT2AMEN1ALDH1A1LMNATHRB
SCHEMBL8643121 0.80 ALDH1A1 (0.59) KMT2AMEN1ALDH1A1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed