SCHEMBL8649485

SCHEMBL8649485

NC(=NO)c1c(Cl)cccc1[AsH2]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
POLB P06746 2/20 0.39
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
HTR3E A5X5Y0 3/20 0.34
HTR3B O95264 3/20 0.34
HTR3A P46098 3/20 0.34
HTR3D Q70Z44 3/20 0.34
HTR3C Q8WXA8 3/20 0.34
ADRA2A P08913 3/20 0.34
HTR1A P08908 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
MAOA P21397 2/20 0.34
ADRA1D P25100 2/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
ADRA1A P35348 2/20 0.34
DRD3 P35462 2/20 0.34
HTR2B P41595 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL102501 0.86 ALDH1A1 (0.50) ALDH1A1POLBGAAGFERHTR3E
SCHEMBL102502 0.86 ALDH1A1 (0.50) ALDH1A1POLBGAAGFERHTR3E
SCHEMBL8381824 0.78 ALDH1A1 (0.43) ALDH1A1POLBGAAGFERHTR3E
SCHEMBL102163 0.77 POLB (0.42) ALDH1A1POLBGAAGFERHTR3E
SCHEMBL102164 0.77 POLB (0.42) ALDH1A1POLBGAAGFERHTR3E
SCHEMBL7242129 0.77 PBRM1 (0.44) ALDH1A1POLBGAATAAR1MEN1
SCHEMBL17737959 0.68 TSHR (0.50) ALDH1A1GAAGFERSMN1; SMN2S100B
SCHEMBL102710 0.68 TSHR (0.50) ALDH1A1GAAGFERSMN1; SMN2S100B
SCHEMBL102709 0.68 TSHR (0.50) ALDH1A1GAAGFERSMN1; SMN2S100B
SCHEMBL101068 0.67 L3MBTL1 (0.50) ALDH1A1POLBGAAGFERHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858451-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-08-19 EP disclosed
WO-1997014686-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS ASTRA PHARMACEUTICALS LIMITED (GB) 1997-04-24 WO disclosed