SCHEMBL8649704

SCHEMBL8649704

O=C1CN(CCCN2CCC(Cc3ccccc3)CC2)S(=O)(=O)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.56
CCR3 P51677 3/20 0.51
SIGMAR1 Q99720 2/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
KCNH2 Q12809 1/20 0.49
MDM2 Q00987 1/20 0.49
KMT2A Q03164 1/20 0.49
CTDSP1 Q9GZU7 1/20 0.49
ADRB2 P07550 1/20 0.48
CHRM2 P08172 1/20 0.48
CHRM4 P08173 1/20 0.48
ADRB1 P08588 1/20 0.48
CHRM5 P08912 1/20 0.48
CHRM1 P11229 1/20 0.48
DRD2 P14416 1/20 0.48
CHRM3 P20309 1/20 0.48
DRD4 P21917 1/20 0.48
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8787330 0.99 TDP1 (0.55) TDP1CCR3SIGMAR1SLC6A2SLC6A4
SCHEMBL8644528 0.93 TDP1 (0.58) TDP1CCR3SIGMAR1MDM2KMT2A
Hydrochloric Acid SCHEMBL8649115 0.92 TDP1 (0.57) TDP1CCR3SIGMAR1MDM2KMT2A
SCHEMBL8788275 0.89 OPRM1 (0.49) TDP1SLC6A2SLC6A4KMT2ADRD2
Hydrochloric Acid SCHEMBL8786910 0.88 OPRM1 (0.48) TDP1SLC6A2SLC6A4KMT2ADRD2
SCHEMBL8648331 0.84 TDP1 (0.53) TDP1SIGMAR1MDM2KMT2ACTDSP1
SCHEMBL8644165 0.84 TDP1 (0.68) TDP1MDM2KMT2ACTDSP1
Hydrochloric Acid SCHEMBL8645889 0.83 TDP1 (0.52) TDP1SIGMAR1MDM2KMT2ACTDSP1
Hydrochloric Acid SCHEMBL8643749 0.83 TDP1 (0.67) TDP1MDM2KMT2ACTDSP1
SCHEMBL8648721 0.82 TDP1 (0.49) TDP1MDM2KMT2ACTDSP1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773437-A UROGENITAL DISORDERS SUCH AS DYSURIA NIPPON CHEMIPHAR CO., LTD. (JP) 1998-06-30 US disclosed
EP-0753514-A1 ALKYLENEDIAMINE DERIVATIVE NIPPON CHEMIPHAR CO., LTD. (JP) 1997-01-15 EP disclosed