SCHEMBL8650840

SCHEMBL8650840

N=C(N)NC(=O)/C(=C/c1cccc(C(F)(F)F)c1)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
P4HB P07237 1/20 0.44
TBXAS1 P24557 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
RECQL P46063 1/20 0.42
NAMPT P43490 1/20 0.42
CSF1R P07333 4/20 0.42
BRAF P15056 2/20 0.42
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
VNN1 O95497 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
EPHX2 P34913 1/20 0.40
TBXA2R P21731 1/20 0.40
KIF11 P52732 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8644166 0.85 CYP1A1 (0.52) MEN1KMT2AP4HBKDM4EGAA
SCHEMBL8647943 0.84 CYP1A2 (0.47) MEN1KMT2ANAMPTALOX15NPSR1
SCHEMBL8645267 0.83 CYP1A1 (0.47) MEN1KMT2AKDM4EPOLBGAA
SCHEMBL8645512 0.82 TSHR (0.54) TSHRMEN1KMT2AP4HBTBXAS1
SCHEMBL8645516 0.82 TSHR (0.54) TSHRMEN1KMT2AP4HBTBXAS1
SCHEMBL8648599 0.81 ALDH1A1 (0.42) MEN1KMT2AP4HBRECQLBRAF
SCHEMBL8648534 0.81 CYP1A1 (0.55) TSHRMEN1KMT2APOLBMAPT
SCHEMBL8649085 0.80 LMNA (0.44) MEN1KMT2ARECQLBRAFMAPT
SCHEMBL8646691 0.80 CYP1A1 (0.47) KMT2AP4HBNAMPTKDM4EGAA
SCHEMBL8650818 0.80 NAMPT (0.46) NAMPTBRAFVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed