SCHEMBL8650842

SCHEMBL8650842

CS(=O)(=O)c1ccccc1/C=C(/C(=O)O)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.46
AKR1C2 P52895 1/20 0.46
AKR1C1 Q04828 1/20 0.46
ALDH1A1 P00352 2/20 0.43
APP P05067 1/20 0.43
GAA P10253 1/20 0.43
HCAR3 P49019 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
AKR1C3 P42330 1/20 0.43
PLOD2 O00469 1/20 0.41
CYP3A4 P08684 3/20 0.41
CYP1A1 P04798 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1B1 Q16678 2/20 0.41
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650850 1.00 PTGS2 (0.46) PTGS2AKR1C2AKR1C1ALDH1A1APP
SCHEMBL8650946 0.82 F7 (0.38) PTGS2ALDH1A1PLOD2CYP3A4CYP1A1
SCHEMBL8643722 0.81 ALDH1A1 (0.47) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8643718 0.81 ALDH1A1 (0.47) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8648115 0.79 ALDH1A1 (0.60) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8648112 0.79 ALDH1A1 (0.60) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8648199 0.79 ALDH1A1 (0.47) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8648195 0.79 ALDH1A1 (0.47) AKR1C1ALDH1A1APPGAAHCAR3
SCHEMBL8646768 0.78 CYP1A1 (0.63) ALDH1A1GAACYP3A4CYP1A1CYP1A2
SCHEMBL8646765 0.78 CYP1A1 (0.63) ALDH1A1GAACYP3A4CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed