SCHEMBL8651256

SCHEMBL8651256

CCCCCCCCc1cccc(C(C=C(C)C)SC(C=C(C)C)c2cccc(CCCCCCCC)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPL P06858 2/20 0.47
LIPG Q9Y5X9 2/20 0.47
PPARA Q07869 2/20 0.43
DRD2 P14416 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
PPARG P37231 1/20 0.41
ESR1 P03372 2/20 0.41
ADRA2A P08913 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
TACR2 P21452 2/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
PTGS2 P35354 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560062 1.00 LPL (0.47) LPLLIPGPPARADRD2OPRM1
SCHEMBL8564542 0.99 LPL (0.46) LPLLIPGPPARADRD2OPRM1
SCHEMBL8564062 0.94 LPL (0.40) LPLLIPGPPARADRD2OPRM1
SCHEMBL8565354 0.89 DRD2 (0.36) DRD2OPRM1DRD3OPRD1OPRK1
SCHEMBL2464423 0.75 LPL (0.54) LPLLIPGPPARADRD2OPRM1
SCHEMBL9835921 0.74 LPL (0.54) LPLLIPGPPARAPPARG
SCHEMBL22795880 0.73 LPL (0.53) LPLLIPGPPARADRD2OPRM1
SCHEMBL27657598 0.73 LPL (0.53) LPLLIPGPPARADRD2OPRM1
Hydrochloric Acid SCHEMBL28356096 0.73 PTGS2 (0.63) LPLLIPGDRD2OPRM1DRD3
SCHEMBL10235993 0.73 LPL (0.53) LPLLIPGPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0568898-B1 Benzothiepine-, benzothiopyrane- and benzothiophenyle derivatives, their preparation and use as medicine HOFFMANN LA ROCHE (CH) 1998-04-01 EP disclosed
EP-0568898-A1 Benzothiepine-, benzothiopyrane- and benzothiophenyle derivatives, their preparation and use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1993-11-10 EP disclosed