SCHEMBL8653003

SCHEMBL8653003

O=C(C#Cc1ccccc1)c1ccc(Cl)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
TSHR P16473 1/20 0.53
CASP1 P29466 1/20 0.53
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
HIF1A Q16665 1/20 0.49
ERCC5 P28715 1/20 0.47
FEN1 P39748 1/20 0.47
FLT1 P17948 2/20 0.46
FLT4 P35916 2/20 0.46
KDR P35968 2/20 0.46
AKR1C2 P52895 1/20 0.45
AKR1C1 Q04828 1/20 0.45
VCP P55072 1/20 0.45
RAB9A P51151 7/20 0.45
NPC1 O15118 6/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
TDP1 Q9NUW8 1/20 0.45
SRD5A2 P31213 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29693880 0.84 NPC1 (0.43) SMN1; SMN2ALDH1A1AKR1C2AKR1C1VCP
SCHEMBL8653177 0.83 ALDH1A1 (0.53) SMN1; SMN2TSHRALDH1A1ERCC5FEN1
SCHEMBL20512347 0.82 SMN1; SMN2 (0.63) SMN1; SMN2TSHRCASP1ALDH1A1MAPK1
SCHEMBL28687224 0.81 VCP (0.43) SMN1; SMN2TSHRCASP1ALDH1A1AKR1C2
SCHEMBL28173510 0.81 SMN1; SMN2 (0.44) SMN1; SMN2TSHRCASP1ALDH1A1MAPK1
SCHEMBL28141856 0.80 SMN1; SMN2 (0.60) SMN1; SMN2TSHRCASP1ALDH1A1MAPK1
SCHEMBL27167237 0.79 CES2 (0.43) ALDH1A1HSP90AA1MAPTPTGDR2
SCHEMBL8652597 0.76 VCP (0.69) SMN1; SMN2TSHRALDH1A1VCPRAB9A
SCHEMBL7202005 0.76 SMN1; SMN2 (0.50) SMN1; SMN2TSHRCASP1ALDH1A1MAPK1
SCHEMBL29625166 0.75 NPC1 (0.55) SMN1; SMN2ALDH1A1AKR1C2AKR1C1VCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1228076-A Diaryl acetylene ketones BAYER AG (DE) 1999-09-08 CN disclosed
EP-0866785-A1 DIARYL ACETYLENE KETONES BAYER AG (DE) 1998-09-30 EP disclosed
WO-1997021658-A1 DIARYL ACETYLENE KETONES BAYER AKTIENGESELLSCHAFT (DE) 1997-06-19 WO disclosed