SCHEMBL8654530

SCHEMBL8654530

CCCCc1c(-c2ccc(O)cc2)oc2c1C(=O)CC(O)=C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.37
ESR1 P03372 7/20 0.36
ESR2 Q92731 7/20 0.36
PPARG P37231 1/20 0.36
CCNB2 O95067 1/20 0.34
CCNE2 O96020 1/20 0.34
INSR P06213 1/20 0.34
CDK1 P06493 1/20 0.34
CFTR P13569 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
MAPK3 P27361 1/20 0.34
MAPK1 P28482 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
MAPK10 P53779 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8656916 0.93 ESR1 (0.42) PTPN1ESR1ESR2PPARGCCNB2
SCHEMBL8657893 0.88 ESR1 (0.47) PTPN1ESR1ESR2MAPK1ALDH1A1
SCHEMBL8653867 0.73 PTPN1 (0.36) PTPN1ESR1ESR2PPARGCCNB2
SCHEMBL8637350 0.65 ALDH1A1 (0.53) PTPN1PPARGMAPK1HSD17B3ALDH1A1
SCHEMBL8638111 0.65 MEN1 (0.51) PTPN1PPARGMAPK1ALOX5HSD17B3
SCHEMBL8653155 0.65 ESR1 (0.39) PTPN1ESR1ESR2PPARGCCNB2
SCHEMBL25144838 0.62 ELANE (0.44) MAPK1ALOX5ALDH1A1GAAABCB1
SCHEMBL25144976 0.60 ELANE (0.44) MAPK1HSD17B3ALDH1A1GAA
SCHEMBL7371867 0.59 TERT (0.64) PTPN1ESR1ESR2MAPK1CDK5
SCHEMBL18770769 0.58 TYR (0.49) PTPN1ESR1ESR2CCNB2CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0516257-B1 Phenylbenzo[b]furans and -thiophenes, procedures for their preparation, and pharmaceutical compositions containing the same SCHERING AG (DE) 1998-08-05 EP claimed