SCHEMBL8655558

SCHEMBL8655558

Cc1csc(C(=O)C2C(=O)Nc3ccc(Cl)nc32)c1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.36
KDR P35968 3/20 0.35
CASP3 P42574 2/20 0.35
SENP7 Q9BQF6 2/20 0.35
CCR2 P41597 2/20 0.33
SENP8 Q96LD8 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
KDM5A P29375 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27408530 0.89 KDR (0.32) KDRCASP3SENP7CCR2DRD2
SCHEMBL27309302 0.80
SCHEMBL8657477 0.80 TDP1 (0.37) DAO
SCHEMBL8654616 0.79 DAO (0.36) DAOKDRCASP3SENP7KDM5A
Ammonia Solution, Strong SCHEMBL27320686 0.79 TDP1 (0.36) DAO
SCHEMBL27363938 0.75 GAA (0.36)
SCHEMBL8653988 0.74 DAO (0.36) DAOKDM5A
SCHEMBL8653164 0.74 DAO (0.34) DAOKDRCASP3SENP7CCR2
SCHEMBL8657361 0.74 HTT (0.41)
SCHEMBL25898804 0.72 MEN1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811432-A Azaoxindole derivatives PFIZER INC (US) 1998-09-22 US disclosed
CN-1031053-C Azaoxindole derivatives PFIZER (US) 1996-02-21 CN disclosed
CN-1053065-A AZAOXINDOLE DERIVATIVES PFIZER (US) 1991-07-17 CN disclosed
WO-1991009598-A1 AZAOXINDOLE DERIVATIVES PFIZER INC. (US) 1991-07-11 WO disclosed
EP-0436333-A2 Azaoxindole derivatives PFIZER INC. (US) 1991-07-10 EP disclosed