SCHEMBL8653164

SCHEMBL8653164

Cc1csc(C(=O)C2C(=O)N(C(N)=O)c3ccc(Cl)nc32)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.34
KDR P35968 3/20 0.33
CASP3 P42574 2/20 0.33
SENP7 Q9BQF6 2/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
KDM5A P29375 1/20 0.31
CCR2 P41597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8653298 0.89
SCHEMBL8657517 0.81 HSD17B10 (0.35) DAO
SCHEMBL8654029 0.77 DAO (0.33) DAOKDM5A
SCHEMBL27408529 0.77 KDR (0.32) KDRCASP3SENP7
SCHEMBL8654034 0.76 EP300 (0.40)
SCHEMBL8655558 0.74 DAO (0.36) DAOKDRCASP3SENP7SENP8
SCHEMBL7885934 0.72 CASP3 (0.38) CASP3
SCHEMBL8652706 0.72 ALDH1A1 (0.36)
SCHEMBL7894075 0.71 CES2 (0.34)
SCHEMBL7895781 0.71 GSK3B (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811432-A Azaoxindole derivatives PFIZER INC (US) 1998-09-22 US claimed
EP-0436333-A2 Azaoxindole derivatives PFIZER INC. (US) 1991-07-10 EP claimed
US-5811432-A Azaoxindole derivatives PFIZER INC (US) 1998-09-22 US disclosed
CN-1053065-A AZAOXINDOLE DERIVATIVES PFIZER (US) 1991-07-17 CN disclosed
WO-1991009598-A1 AZAOXINDOLE DERIVATIVES PFIZER INC. (US) 1991-07-11 WO disclosed
EP-0436333-A2 Azaoxindole derivatives PFIZER INC. (US) 1991-07-10 EP disclosed