SCHEMBL8660844

SCHEMBL8660844

Cc1cc(Oc2ccc(Br)cc2Br)c(Cl)c(C)c1NC(=O)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
ATM Q13315 1/20 0.40
KDM4E B2RXH2 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GHSR Q92847 1/20 0.36
KMT2A Q03164 3/20 0.36
EPAS1 Q99814 1/20 0.36
MEN1 O00255 1/20 0.35
MAPK1 P28482 2/20 0.35
PYGL P06737 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HDAC1 Q13547 1/20 0.35
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660840 0.96 MAPT (0.40) MAPTPOLBATMKDM4ERXFP1
SCHEMBL8658883 0.94 MEN1 (0.41) MAPTPOLBATMKDM4EKMT2A
SCHEMBL8662538 0.92 MAPT (0.41) MAPTPOLBATMGHSRKMT2A
SCHEMBL8662521 0.90 ALDH1A1 (0.39) MAPTPOLBKDM4ERXFP1KMT2A
SCHEMBL27694017 0.90 MAPT (0.43) MAPTPOLBATMGHSRKMT2A
SCHEMBL8656117 0.89 PYGL (0.48) MAPTPOLBGHSRKMT2AMEN1
SCHEMBL8663050 0.86 MEN1 (0.41) MAPTPOLBATMKDM4EKMT2A
SCHEMBL8656588 0.85 GCGR (0.42) MAPTPOLBATMGHSRKMT2A
SCHEMBL8660976 0.85 MAPT (0.40) MAPTPOLBATMPYGLALDH1A1
SCHEMBL8659406 0.84 KMT2A (0.42) MAPTKDM4ERXFP1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed