SCHEMBL8656182

SCHEMBL8656182

NS(=O)(=O)c1ccccc1-c1cc2c(cc1-c1cc(Cl)c(C(F)(F)F)c(Cl)c1)OCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.38
PTGS1 P23219 4/20 0.38
F10 P00742 4/20 0.37
PTGES2 Q9H7Z7 1/20 0.37
FABP4 P15090 1/20 0.35
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
PTPRC P08575 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657920 0.87 PTGS2 (0.44) PTGS2PTGS1F10CA12CA2
SCHEMBL8656159 0.87 PTGS2 (0.43) PTGS2PTGS1F10PTGES2CA12
SCHEMBL8661240 0.87 PTGS2 (0.42) PTGS2PTGS1F10PTGES2CA12
SCHEMBL8659133 0.87 FABP4 (0.45) PTGS2PTGS1F10PTGES2FABP4
SCHEMBL8656123 0.86 F10 (0.39) PTGS2PTGS1F10CA12CA2
SCHEMBL8661053 0.85 PTGS2 (0.40) PTGS2PTGS1F10PTGES2CA12
SCHEMBL8656674 0.84 PTGS2 (0.45) PTGS2PTGS1F10PTGES2ALOX5AP
SCHEMBL8657983 0.84 PTGS2 (0.45) PTGS2PTGS1PTGES2CA12CA2
SCHEMBL8661927 0.84 PTGS2 (0.36) PTGS2PTGS1F10CA12CA2
SCHEMBL8662987 0.83 PTGS2 (0.46) PTGS2PTGS1F10CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed