SCHEMBL8657152

SCHEMBL8657152

Cc1cc(NC(=O)NC(=O)c2c(F)cccc2F)c(C)c(Cl)c1Oc1cccc(-c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
MAPT P10636 3/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
ATM Q13315 1/20 0.40
IL2 P60568 1/20 0.37
RAB9A P51151 3/20 0.36
DHODH Q02127 2/20 0.36
POLB P06746 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
VCP P55072 1/20 0.36
NPC1 O15118 1/20 0.35
PYGL P06737 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
THRB P10828 1/20 0.35
RECQL P46063 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660055 0.88 KMT2A (0.53) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL9135516 0.87 MEN1 (0.52) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8656618 0.87 MEN1 (0.44) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8660974 0.86 KMT2A (0.47) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8657367 0.84 KMT2A (0.51) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8664786 0.84 MEN1 (0.45) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8659761 0.84 MEN1 (0.45) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8659824 0.83 MEN1 (0.47) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8665574 0.82 KMT2A (0.51) MEN1KMT2AMAPTUSP2ALOX15
SCHEMBL8661518 0.82 MEN1 (0.47) MEN1KMT2AMAPTUSP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0186297-B1 PESTICIDAL BIPHENYLYLOXY AND BIPHENYLYLALKOXY ARYL ACYL UREA COMPOUNDS, A PROCESS FOR THEIR PREPARATION, PESTICIDAL COMPOSITIONS AND A METHOD OF CONTROLLING PESTS RHONE-POULENC NEDERLAND B.V. (NL) 1989-03-08 EP disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
US-4638088-A INSECTICIDES, MITICIDES UNION CARBIDE CORPORATION (US) 1987-01-20 US disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0186297-A1 Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds, a process for their preparation, pesticidal compositions and a method of controlling pests RHONE-POULENC NEDERLAND B.V. (NL) 1986-07-02 EP disclosed