SCHEMBL8660974

SCHEMBL8660974

Cc1cc(NC(=O)NC(=O)c2c(F)cccc2F)c(C)c(Cl)c1Oc1ccccc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
MAPT P10636 2/20 0.42
USP2 O75604 1/20 0.42
ALOX15 P16050 1/20 0.42
ATM Q13315 2/20 0.41
GCK P35557 1/20 0.40
PPIA P62937 3/20 0.40
SCN9A Q15858 1/20 0.39
PYGL P06737 2/20 0.39
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
RECQL P46063 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 1/20 0.38
DHODH Q02127 1/20 0.37
IL2 P60568 1/20 0.37
DYRK3 O43781 1/20 0.36
PRKD3 O94806 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660963 0.95 PPIA (0.46) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8657024 0.95 KMT2A (0.45) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8664786 0.92 MEN1 (0.45) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8659761 0.92 MEN1 (0.45) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL10599956 0.91 PYGL (0.49) KMT2AMAPTPPIASCN9APYGL
SCHEMBL8657367 0.89 KMT2A (0.51) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8661107 0.88 MEN1 (0.43) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8656985 0.88 MEN1 (0.41) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8657152 0.86 MEN1 (0.47) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL8656618 0.86 MEN1 (0.44) KMT2AMEN1MAPTUSP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186297-B1 PESTICIDAL BIPHENYLYLOXY AND BIPHENYLYLALKOXY ARYL ACYL UREA COMPOUNDS, A PROCESS FOR THEIR PREPARATION, PESTICIDAL COMPOSITIONS AND A METHOD OF CONTROLLING PESTS RHONE-POULENC NEDERLAND B.V. (NL) 1989-03-08 EP claimed
US-4638088-A INSECTICIDES, MITICIDES UNION CARBIDE CORPORATION (US) 1987-01-20 US claimed
EP-0186297-A1 Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds, a process for their preparation, pesticidal compositions and a method of controlling pests RHONE-POULENC NEDERLAND B.V. (NL) 1986-07-02 EP claimed
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
US-4638088-A INSECTICIDES, MITICIDES UNION CARBIDE CORPORATION (US) 1987-01-20 US disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0186297-A1 Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds, a process for their preparation, pesticidal compositions and a method of controlling pests RHONE-POULENC NEDERLAND B.V. (NL) 1986-07-02 EP disclosed