SCHEMBL8658024

SCHEMBL8658024

CN(C)c1cc(N(c2ccccc2)S(=O)(=O)c2ccccc2)cc(N(C)C)c1F

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.51
ESR1 P03372 1/20 0.49
HTR6 P50406 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 3/20 0.40
NR1H3 Q13133 3/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 1/20 0.38
HSD11B1 P28845 1/20 0.37
NR1H2 P55055 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8659118 0.89 PKM (0.53) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8663371 0.86 PKM (0.53) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8658102 0.85 PKM (0.49) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8659634 0.85 PKM (0.51) PKMESR1HTR6CA12CA9
SCHEMBL8659111 0.84 PKM (0.47) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8659120 0.82 PKM (0.49) PKMESR1HTR6CA12CA9
SCHEMBL8656891 0.82 PKM (0.49) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8658317 0.82 PKM (0.59) PKMESR1APOBEC3GCA12CA9
SCHEMBL8656901 0.82 PKM (0.51) PKMESR1HTR6APOBEC3GCA12
SCHEMBL8660081 0.81 PKM (0.50) PKMESR1HTR6CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed