SCHEMBL8658317

SCHEMBL8658317

CN(C)c1cc(N(C)C)cc(N(c2ccccc2)S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.59
ESR1 P03372 1/20 0.56
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
ALDH1A1 P00352 4/20 0.44
APOBEC3G Q9HC16 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD11B1 P28845 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
NR1H3 Q13133 1/20 0.41
NR1I2 O75469 1/20 0.41
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8663009 0.91 PKM (0.58) PKMESR1CA12CA9ALDH1A1
SCHEMBL8656925 0.89 PKM (0.63) PKMESR1CA12CA9ALDH1A1
SCHEMBL8660142 0.85 PKM (0.54) PKMESR1CA12CA9ALDH1A1
SCHEMBL812682 0.84 PKM (0.79) PKMESR1CA12CA9ALDH1A1
SCHEMBL8663371 0.83 PKM (0.53) PKMESR1CA12CA9ALDH1A1
SCHEMBL8659118 0.83 PKM (0.53) PKMESR1CA12CA9ALDH1A1
SCHEMBL8656901 0.82 PKM (0.51) PKMESR1CA12CA9ALDH1A1
SCHEMBL8658024 0.82 PKM (0.51) PKMESR1CA12CA9ALDH1A1
SCHEMBL8658027 0.82 PKM (0.51) PKMESR1CA12CA9ALDH1A1
SCHEMBL8659634 0.82 PKM (0.51) PKMESR1CA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed