SCHEMBL8658182

SCHEMBL8658182

CCCC(=O)Oc1ccc(C#Cc2cc3c(cc2C)OCCC3(CC)CC)o1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
MAP3K14 Q99558 1/20 0.32
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664152 0.91 MAP3K14 (0.32) MAP3K14
SCHEMBL8663440 0.88 MAP3K14 (0.30) MAP3K14
SCHEMBL8661859 0.84 PTGS2 (0.31)
SCHEMBL8663438 0.84 KDM4E (0.31) KDM4EALDH1A1GLAGAAKMT2A
SCHEMBL8659864 0.82
SCHEMBL8660965 0.82 KMT2A (0.35) KDM4EALDH1A1GLAGAAKMT2A
SCHEMBL8658185 0.81 NPC1 (0.31) ALDH1A1GLAPRSS1PRSS2PRSS3
SCHEMBL8661130 0.81
SCHEMBL8663221 0.80 KMT2A (0.34) KDM4EALDH1A1GLAGAAKMT2A
SCHEMBL7654818 0.80 PRSS1 (0.33) MAP3K14PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed