SCHEMBL8658481

SCHEMBL8658481

CN1CCCCC1CCc1cc2c(cc1Br)CCN2C(=O)Nc1ccc(-c2ccncc2)c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.55
HTR1D P28221 1/20 0.55
HTR1B P28222 1/20 0.55
HTR2C P28335 7/20 0.41
HTR2A P28223 6/20 0.41
HTR2B P41595 3/20 0.41
DRD1 P21728 1/20 0.41
HRH2 P25021 1/20 0.41
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41
CHRM3 P20309 10/20 0.40
POLB P06746 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618345 0.84 HTR1A (0.62) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8613994 0.82 HTR1A (0.57) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8128883 0.79 HTR1A (0.64) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8127323 0.78 HTR1A (0.81) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8618094 0.77 HTR1A (0.62) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8620951 0.76 TSHR (0.42) HTR2CHTR2AHTR2BDRD1HRH2
SCHEMBL8122308 0.75 HTR1A (0.73) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8128007 0.74 HTR1A (0.79) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8614116 0.73 HTR1D (0.57) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8137992 0.73 HTR1A (0.72) HTR1AHTR1DHTR1BHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed