SCHEMBL8658685

SCHEMBL8658685

Cc1ccc2[nH]cc(Cc3cccnc3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
PCSK9 Q8NBP7 1/20 0.51
HTR1D P28221 4/20 0.50
HTR2A P28223 2/20 0.50
MAP2K4 P45985 1/20 0.47
SNCA P37840 1/20 0.47
IDO1 P14902 1/20 0.45
GABRA1 P14867 1/20 0.45
GABRB2 P47870 1/20 0.45
HTR1B P28222 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SPR P35270 1/20 0.44
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MET P08581 1/20 0.43
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
DRD2 P14416 1/20 0.42
ADRA2B P18089 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540445 0.84 GPR84 (0.63) HTR1DHTR2ASNCAIDO1GABRA1
SCHEMBL5725721 0.84 GPR84 (0.63) HTR2AKMT2AHTR1ASLC6A4
SCHEMBL8657374 0.84 GPR84 (0.63) PCSK9HTR2ASNCAIDO1KMT2A
SCHEMBL8658847 0.83 GPR84 (0.66) HTR1DHTR2AHTR1BMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL8658852 0.82 GPR84 (0.64) HTR1DHTR2AHTR1BMTNR1AMTNR1B
SCHEMBL5870915 0.81 MEN1 (0.68) MEN1KMT2AMETHTR6
SCHEMBL8656583 0.81 SLC6A4 (0.48) SNCAHTR1ADRD2SLC6A4DRD3
SCHEMBL14194176 0.80 CYP3A4 (0.60) MET
SCHEMBL18383116 0.79 HTR1D (0.69) PCSK9HTR1DHTR2AHTR1BMEN1
SCHEMBL8541224 0.79 CYP19A1 (0.53) GAASNCAGABRA1GABRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834493-A TREATMENT OF NERVOUS SYSTEM DISORDERS GIL QUINTERO MYRNA (IT) 1998-11-10 US disclosed
CN-1124960-A Indole derivatives as 5-HT1A and/or 5-HT2 ligands BOEHRINGER INGELHEIM ITALIA (IT) 1996-06-19 CN disclosed
EP-0694033-A1 INDOLE DERIVATIVES AS 5-HT1A AND/OR 5-HT2 LIGANDS BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1996-01-31 EP disclosed
WO-1994024125-A1 INDOLE DERIVATIVES AS 5-HT1A AND/OR 5-HT2 LIGANDS BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1994-10-27 WO disclosed