SCHEMBL8660079

SCHEMBL8660079

C=Cc1c(Br)cc([N+](=O)[O-])c(N)c1CNC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
CYP3A4 P08684 1/20 0.39
CTSB P07858 1/20 0.38
POLB P06746 2/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 6/20 0.32
PKM P14618 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
KMT2A Q03164 2/20 0.31
LMNA P02545 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
G6PD P11413 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
CYP2D6 P10635 1/20 0.31
GAA P10253 1/20 0.31
CA12 O43570 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660076 0.81 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSBPOLBHTT
SCHEMBL7566874 0.74 GRIA1 (0.42) ALDH1A1CYP3A4CTSBPOLBHTT
SCHEMBL27486507 0.73 GRIA1 (0.34) ALDH1A1CYP3A4CTSBPOLBHTT
SCHEMBL27436503 0.71 GRIA1 (0.33) ALDH1A1CYP3A4CTSBPOLBPKM
SCHEMBL7566388 0.71 GRIA1 (0.49) ALDH1A1HTTMAPTKMT2ALMNA
SCHEMBL8640535 0.68 TSHR (0.45) ALDH1A1CYP3A4MAPTTDP1KMT2A
SCHEMBL31248962 0.67 HPGD (0.39) ALDH1A1CYP3A4POLBMAPTTDP1
SCHEMBL19643097 0.66 TDP1 (0.44) ALDH1A1CYP3A4POLBMAPTTDP1
SCHEMBL7572511 0.65 GRIA1 (0.59) ALDH1A1KMT2AKDM4EMEN1
SCHEMBL28385538 0.65 ALDH1A1 (0.49) ALDH1A1CYP3A4POLBHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1125818-C Amino acid derivatives of substituted quinoxaline 2, 3 -dione derivativesa as glutamate receptor antagonists WARNER LAMBERT CO (US) 2003-10-29 CN disclosed
EP-0832074-A1 AMINO ACID DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONE DERIVATIVES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-04-01 EP disclosed