SCHEMBL8660189

SCHEMBL8660189

COc1cc(OC)cc(-c2ccccc2-c2ccccc2S(N)(=O)=O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.56
ABCB1 P08183 2/20 0.56
BCR P11274 2/20 0.56
PTGES2 Q9H7Z7 1/20 0.46
P2RX3 P56373 1/20 0.45
USP2 O75604 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
KMT2A Q03164 1/20 0.42
PTGS2 P35354 3/20 0.42
PTGS1 P23219 2/20 0.42
SCN9A Q15858 1/20 0.41
F10 P00742 4/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657999 0.88 PTGES2 (0.56) PTGES2PTGS2PTGS1F10CA1
SCHEMBL8659255 0.87 ABL1 (0.45) ABL1ABCB1BCRPTGES2P2RX3
SCHEMBL8662983 0.86 SCN9A (0.53) ABL1ABCB1BCRPTGES2MAPT
SCHEMBL8661454 0.83 ABL1 (0.41) ABL1ABCB1BCRPTGES2P2RX3
SCHEMBL8658511 0.82 PTGS2 (0.40) PTGES2PTGS2PTGS1F10CYP2C9
SCHEMBL8656781 0.82 CA9 (0.54) MAPTKMT2APTGS2PTGS1CA1
SCHEMBL8661248 0.82 PTGS2 (0.46) PTGES2USP2MAPTPKMKMT2A
SCHEMBL6725549 0.81 ABL1 (0.65) ABL1ABCB1BCRPTGS2PTGS1
SCHEMBL4662753 0.81 PTGES2 (0.59) PTGES2P2RX3F10CA1CA2
SCHEMBL8663003 0.81 PTGS2 (0.51) PTGES2USP2MAPTPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed