SCHEMBL8660682

SCHEMBL8660682

c1cc2occc2cn1.c1ccc2c(c1)CC2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.41
CYP11B2 P19099 10/20 0.37
CYP11B1 P15538 9/20 0.37
CYP19A1 P11511 7/20 0.37
SIGMAR1 Q99720 1/20 0.37
NAMPT P43490 1/20 0.36
CYP17A1 P05093 1/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
EED O75530 1/20 0.33
NPY5R Q15761 1/20 0.33
CYP3A4 P08684 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL88833 0.85
SCHEMBL29813261 0.85
SCHEMBL15971546 0.83 DYRK1A (0.50) DYRK1ANAMPTCYP3A4KDM4EALDH1A1
Isoquinoline SCHEMBL10682580 0.75 DYRK1A (0.43) DYRK1ACYP11B2CYP11B1CYP19A1NAMPT
Benzofuran SCHEMBL20488656 0.71 TSHR (0.46) NPY5RSLC6A2SLC6A4SLC6A3
SCHEMBL31692910 0.69 ALDH1A1 (0.38) DYRK1ACYP11B2CYP11B1CYP19A1NAMPT
SCHEMBL10824 0.69
Benzofuran SCHEMBL11554408 0.67 DYRK1A (0.50) DYRK1ANAMPTALDH1A1
Isoquinoline SCHEMBL9777562 0.67 SIGMAR1 (0.57) CYP11B2CYP11B1CYP19A1SIGMAR1CHRNB2
SCHEMBL32685371 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770763-A POLYARYLCYCLOBUTENES DERIVED FROM 3,6 FUNCTIONALIZED MONO AND DICYCLOBUTABENZENE THE BOARD OF REGENTS OF THE UNIV. OF MICHIGAN (US) 1998-06-23 US disclosed
US-5552508-A Difunctional bitricyclodecatriene monomers UNIVERSITY OF MICHIGAN, THE BOARD OF REGENTS (US) 1996-09-03 US disclosed
US-5418312-A Polymer properties THE BOARD OF REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1995-05-23 US disclosed
US-5334752-A Difunctionalized to be incorporated into polymers for compressive strength THE BOARD OF REGENTS ACTING FOR AND ON BEHALF OF UNIVERSITY OF MICHIGAN (US) 1994-08-02 US disclosed
WO-1994001388-A1 CYCLOBUTABENZENE MONOMERS AND METHODS OF MAKING AND USING SAME UNIVERSITY OF MICHIGAN (US) 1994-01-20 WO disclosed