SCHEMBL8660896

SCHEMBL8660896

Cc1cc(NC(=O)NC(=O)c2c(F)cccc2F)ccc1Oc1ncc(C#N)cc1C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
THRB P10828 1/20 0.46
RECQL P46063 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MET P08581 3/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
PKM P14618 1/20 0.42
KDR P35968 5/20 0.41
BRAF P15056 2/20 0.41
MAPK14 Q16539 1/20 0.41
LRRK2 Q5S007 6/20 0.40
MAP3K7 O43318 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658727 0.94 KDM4E (0.47) KDM4EMEN1GAAMAPTTHRB
SCHEMBL8665373 0.92 MEN1 (0.46) KDM4EMEN1GAAMAPTTHRB
SCHEMBL8663074 0.89 TAS1R3 (0.44) KDM4EMEN1KMT2ANPC1KDR
SCHEMBL8659341 0.89 KDM4E (0.47) KDM4EMEN1GAAMAPTTHRB
SCHEMBL10638961 0.85 KDM4E (0.41) KDM4EMEN1GAAMAPTTHRB
SCHEMBL8658837 0.83 TAS1R3 (0.44) KDM4EMEN1MAPTKMT2ANPC1
SCHEMBL8660946 0.83 GCGR (0.51) MEN1KMT2ATDP1NPC1RAB9A
SCHEMBL8659922 0.82 MET (0.42) KDM4EMEN1GAAMAPTTHRB
SCHEMBL8662523 0.81 KDM4E (0.50) KDM4EMEN1GAAMAPTTHRB
SCHEMBL8656206 0.79 KDM4E (0.46) KDM4EMEN1GAAMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
US-4659724-A Certain 1-[4-(5-cyano-2-pyridyloxy)phenyl-benzoyl ureas having pesticidal properties UNION CARBIDE CORPORATION (US) 1987-04-21 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0115210-A1 Pesticidal benzoyl ureas and process for their preparation UNION CARBIDE CORPORATION (US) 1984-08-08 EP disclosed