SCHEMBL8661901

SCHEMBL8661901

CC1c2cc(Br)ccc2OC(C)(C)C1(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.35
PBRM1 Q86U86 1/20 0.34
BACE1 P56817 2/20 0.34
LMNA P02545 2/20 0.33
MAPK1 P28482 1/20 0.33
HTR2B P41595 7/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
PGR P06401 1/20 0.31
ALDH1A1 P00352 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HTT P42858 1/20 0.31
AKR1B1 P15121 1/20 0.31
POLB P06746 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL570350 0.79 MAPT (0.37) HTR2BALDH1A1
SCHEMBL9765072 0.77 ABCB1 (0.34)
SCHEMBL9443650 0.76 LMNA (0.35) AHRPBRM1BACE1LMNAMAPK1
SCHEMBL9872032 0.74 KDM4E (0.39) AKR1B1
SCHEMBL3894061 0.74 KCNE1 (0.35) LMNAHTR2BALDH1A1NPSR1HTT
Arsenic SCHEMBL8675880 0.73 LMNA (0.34) LMNAHTR2BNPSR1HTTTSHR
SCHEMBL9141916 0.71 HTR2A (0.36) AHRLMNAMAPK1HTR2BHTR2A
SCHEMBL23362474 0.70 AHR (0.36) AHRPBRM1BACE1LMNAMAPK1
SCHEMBL11000607 0.70 KCNE1 (0.37) AHRLMNAMAPK1PGRALDH1A1
SCHEMBL29804528 0.70 AHR (0.36) AHRPBRM1BACE1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876330-A1 ARYL OR HETEROARYL AMIDES OF TETRAHYDRONAPHTHALENE, CHROMAN, THIOCHROMAN AND 1,2,3,4-TETRAHYDROQUINOLINE CARBOXYLIC ACIDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1998-11-11 EP disclosed
WO-1997019052-A1 ARYL OR HETEROARYL AMIDES OF TETRAHYDRONAPHTHALENE, CHROMAN, THIOCHROMAN AND 1,2,3,4-TETRAHYDROQUINOLINE CARBOXYLIC ACIDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1997-05-29 WO disclosed