SCHEMBL8662406

SCHEMBL8662406

CCN(CC)CCC1C(=O)C(NC(=O)Nc2ccccc2)[N+](=O)N(CC2CCCCC2)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 5/20 0.40
EPHX1 P07099 2/20 0.39
EPHX2 P34913 3/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ICMT O60725 1/20 0.35
ALB P02768 1/20 0.35
CTSD P07339 1/20 0.34
BACE1 P56817 1/20 0.34
NPC1 O15118 1/20 0.34
ACHE P22303 1/20 0.34
CCKAR P32238 1/20 0.34
CACNA1G O43497 1/20 0.33
CACNA1H O95180 1/20 0.33
CACNA1I Q9P0X4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662408 0.72 CCKBR (0.42) CCKBREPHX1EPHX2RAB9ASMN1; SMN2
SCHEMBL8561164 0.71 CCKBR (0.59) CCKBR
SCHEMBL8866205 0.69 CCKBR (0.51) CCKBR
SCHEMBL8559320 0.69 CCKBR (0.49) CCKBR
SCHEMBL7738117 0.66 CCKBR (0.47) CCKBR
SCHEMBL8563328 0.63 CCKBR (0.49) CCKBR
SCHEMBL8648076 0.62 CCKBR (0.64) CCKBRCCKAR
SCHEMBL23432014 0.59 EPHX1 (1.00) EPHX1EPHX2RAB9ASMN1; SMN2NPC1
SCHEMBL12196136 0.59 EPHX1 (1.00) EPHX1EPHX2RAB9ASMN1; SMN2NPC1
SCHEMBL23431981 0.59 EPHX1 (1.00) EPHX1EPHX2RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710230-B1 1,5-BENZODIAZEPINE DERIVATIVES USEFUL AS CCK OR GASTRIN ANTAGONISTS GLAXO WELLCOME SPA (IT) 1998-09-16 EP claimed