SCHEMBL8662937

SCHEMBL8662937

CCOC(=O)C=Cc1c[nH]c2cnc(-n3cncn3)cc12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
CCNC P24863 5/20 0.39
CDK8 P49336 5/20 0.39
CDK19 Q9BWU1 1/20 0.39
PIM1 P11309 1/20 0.39
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DPP4 P27487 1/20 0.35
P2RY12 Q9H244 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660649 0.84 MAPT (0.44) MAPTKDM4EMEN1KMT2AATM
SCHEMBL8781554 0.75 L3MBTL1 (0.36) MAPTKDM4ECCNCCDK8CDK19
SCHEMBL8781556 0.75 L3MBTL1 (0.36) MAPTKDM4ECCNCCDK8CDK19
SCHEMBL8644915 0.71 PIM1 (0.47) MAPTKDM4EMEN1KMT2APIM1
SCHEMBL15245773 0.70 MAPT (0.58) MAPTKDM4EMEN1KMT2AATM
SCHEMBL8424904 0.70 PIM1 (0.46) MAPTKDM4EKMT2APIM1
SCHEMBL28969558 0.69 MAPT (0.56) MAPTKDM4EMEN1KMT2AATM
SCHEMBL4619581 0.68 MEN1 (0.64) MAPTKDM4EMEN1KMT2AATM
SCHEMBL8650036 0.68 HTR1A (0.51) MAPTKDM4EMEN1KMT2APIM1
SCHEMBL4619586 0.68 MEN1 (0.64) MAPTKDM4EMEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807857-A Piperazine, piperidine and tetrahydropyridine derivative of indol-3-alkyl as 5-HT1D-α agonists MERCK SHARP & DOHME LTD. (GB) 1998-09-15 US disclosed