SCHEMBL8663060

SCHEMBL8663060

O=C(NC(=O)c1ccccc1Cl)Nc1cc(Cl)c(Oc2ccc(Cl)c3ccccc23)c(Cl)c1Cl

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYGL P06737 7/20 0.52
GCGR P47871 1/20 0.47
ESRRA P11474 4/20 0.47
POLB P06746 2/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
PNLIP P16233 1/20 0.39
CYP1A2 P05177 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
PLCG2 P16885 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
GHSR Q92847 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8663155 0.91 PYGL (0.45) PYGLGCGRESRRANPC1RAB9A
SCHEMBL8667260 0.87 PYGL (0.53) PYGLGCGRPOLBNPC1PKM
SCHEMBL8657049 0.86 GCGR (0.59) PYGLGCGRPOLBNPC1PKM
SCHEMBL8655821 0.86 GCGR (0.58) PYGLGCGRESRRAPOLBNPC1
SCHEMBL8657774 0.85 MEN1 (0.55) PYGLESRRAPOLBNPC1RAB9A
SCHEMBL8657108 0.84 PYGL (0.51) PYGLGCGRESRRAPOLBNPC1
SCHEMBL8658823 0.83 PYGL (0.50) PYGLGCGRPOLBNPC1PKM
SCHEMBL8659159 0.83 GCGR (0.51) PYGLGCGRPOLBNPC1PKM
SCHEMBL8662597 0.81 GCGR (0.48) PYGLGCGRPOLBNPC1PKM
SCHEMBL10963721 0.81 ESRRA (0.54) PYGLGCGRESRRAPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed