SCHEMBL8659159

SCHEMBL8659159

O=C(NC(=O)c1ccccc1Cl)Nc1cc(Cl)c(Oc2ccc(Cl)cc2Br)c(Cl)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.51
PYGL P06737 11/20 0.50
PNLIP P16233 2/20 0.42
CXCR2 P25025 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
PARP1 P09874 1/20 0.39
PARG Q86W56 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658823 0.92 PYGL (0.50) GCGRPYGLPNLIPNPC1RAB9A
SCHEMBL8662597 0.92 GCGR (0.48) GCGRPYGLPNLIPNPC1RAB9A
SCHEMBL8663057 0.91 LMNA (0.48) GCGRPYGLPNLIPNPC1RAB9A
SCHEMBL8657049 0.91 GCGR (0.59) GCGRPYGLPNLIPNPC1RAB9A
SCHEMBL8658933 0.89 KMT2A (0.42) GCGRPYGLCXCR2POLBMEN1
SCHEMBL8667260 0.85 PYGL (0.53) GCGRPYGLPNLIPNPC1RAB9A
SCHEMBL9135160 0.84 PYGL (0.49) GCGRPYGLPNLIPCXCR2NPC1
SCHEMBL8658554 0.84 KMT2A (0.50) NPC1PKMMEN1KMT2A
SCHEMBL8659648 0.84 MEN1 (0.54) PYGLCXCR2NPC1RAB9APOLB
SCHEMBL8663060 0.83 PYGL (0.52) GCGRPYGLPNLIPNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed