SCHEMBL8663231

SCHEMBL8663231

C#CCC1NC(=S)N(c2ccc(Cl)cc2C)C1=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
GAA P10253 6/20 0.38
MAPT P10636 3/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
TP53 P04637 1/20 0.32
NPC1 O15118 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK14 Q16539 1/20 0.32
GRM1 Q13255 1/20 0.31
GRM4 Q14833 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662875 0.91 GAA (0.40) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL8662891 0.75 GAA (0.43) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL8663213 0.71 GAA (0.40) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL8526108 0.71 ALDH1A1 (0.42) ALDH1A1KDM4E
SCHEMBL8919380 0.68 KMT2A (0.48) ALDH1A1GAAMAPTMEN1KMT2A
SCHEMBL8661557 0.67 GAA (0.44) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL8663642 0.65 GAA (0.46) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL8663372 0.65 ALDH1A1 (0.44) ALDH1A1GAAMAPTMEN1KMT2A
SCHEMBL10704901 0.64 MGLL (0.55) ALDH1A1MAPTRAB9AKDM4ETP53
SCHEMBL11608600 0.64 MEN1 (0.50) ALDH1A1MAPTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876355-A1 2-THIOXO-IMIDAZOLIDIN-4-ONE DERIVATIVES AND THEIR USE FOR INCREASING HDL CHOLESTEROL CONCENTRATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-11-11 EP claimed
WO-1997019932-A1 2-THIOXO-IMIDAZOLIDIN-4-ONE DERIVATIVES AND THEIR USE FOR INCREASING HDL CHOLESTEROL CONCENTRATION AMERICAN HOME PRODUCTS CORPORATION (US) 1997-06-05 WO claimed