SCHEMBL8663783

SCHEMBL8663783

[c]1occ(-c2ccsc2)c1N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.47
PRKDC P78527 4/20 0.46
PIK3CA P42336 4/20 0.46
PIK3CB P42338 3/20 0.46
PIK3CD O00329 1/20 0.46
PIK3CG P48736 3/20 0.45
RIPK1 Q13546 1/20 0.40
GAK O14976 1/20 0.40
MTOR P42345 1/20 0.39
ATR Q13535 1/20 0.38
ATRIP Q8WXE1 1/20 0.38
EPHX2 P34913 1/20 0.36
ADK P55263 1/20 0.35
FLT1 P17948 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664432 0.80 LMNA (0.47) ARPRKDCALDH1A1MAPTHTT
SCHEMBL8663602 0.78 AR (0.48) ARPRKDCPIK3CAPIK3CBPIK3CD
SCHEMBL8664979 0.78 NPC1 (0.48) PRKDCPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL31025635 0.70 AR (0.55) ARPRKDCPIK3CAPIK3CBPIK3CD
SCHEMBL1310274 0.66 PIK3CA (0.59) ARPRKDCPIK3CAPIK3CBPIK3CD
SCHEMBL27743819 0.66 LMNA (0.52) ARPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL2879730 0.64 AR (0.48) ARPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL17009413 0.64 AR (1.00) ARMEN1NPC1ALDH1A1MAPT
SCHEMBL31060119 0.64 PRKDC (1.00) PRKDCPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL8662677 0.63 PIK3CA (0.47) PRKDCPIK3CAPIK3CBPIK3CDPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852006-A N-aminoalkyl-substituted nitrogen-containing six membered heterocyclic compounds NIPPON CHEMIPHAR CO., LTD. (JP) 1998-12-22 US disclosed
US-5574030-A INHIBITING URINARY CONTRACTION, HETEROCYCLIC DIAMINES NIPPON CHEMIPHAR CO., LTD. (JP) 1996-11-12 US disclosed