SCHEMBL8663602

SCHEMBL8663602

[c]1scc(-c2ccsc2)c1N1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.48
PIK3CA P42336 3/20 0.46
PIK3CB P42338 2/20 0.46
PIK3CG P48736 2/20 0.46
PRKDC P78527 4/20 0.45
PIK3CD O00329 1/20 0.44
GAK O14976 1/20 0.41
MTOR P42345 1/20 0.40
RIPK1 Q13546 1/20 0.39
ATR Q13535 1/20 0.38
ATRIP Q8WXE1 1/20 0.38
EPHX2 P34913 1/20 0.37
ADK P55263 1/20 0.36
PIK3R2 O00459 1/20 0.35
LRRK2 Q5S007 1/20 0.35
GAA P10253 1/20 0.35
FLT1 P17948 2/20 0.34
FLT4 P35916 2/20 0.34
KDR P35968 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664502 0.82 AR (0.47) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL8663783 0.78 AR (0.47) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL8662677 0.75 PIK3CA (0.47) PIK3CAPIK3CBPIK3CGPRKDCPIK3CD
SCHEMBL31025635 0.71 AR (0.55) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL1310274 0.67 PIK3CA (0.59) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL27743819 0.67 LMNA (0.52) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL17009413 0.65 AR (1.00) ARGAA
SCHEMBL2879730 0.65 AR (0.48) ARPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL13000164 0.64 PIK3CA (1.00) PIK3CAPIK3CBPIK3CGPRKDCPIK3CD
SCHEMBL13735487 0.63 AR (0.49) ARPIK3CAPIK3CBPIK3CGPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852006-A N-aminoalkyl-substituted nitrogen-containing six membered heterocyclic compounds NIPPON CHEMIPHAR CO., LTD. (JP) 1998-12-22 US disclosed
US-5574030-A INHIBITING URINARY CONTRACTION, HETEROCYCLIC DIAMINES NIPPON CHEMIPHAR CO., LTD. (JP) 1996-11-12 US disclosed