SCHEMBL8664249

SCHEMBL8664249

N#Cc1cc(Cl)c(F)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 3/20 0.39
KHK P50053 1/20 0.38
CYP11B2 P19099 5/20 0.37
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AR P10275 3/20 0.33
VCAM1 P19320 1/20 0.33
CYP11B1 P15538 2/20 0.33
EGLN2 Q96KS0 1/20 0.33
GRM5 P41594 1/20 0.31
PGK1 P00558 1/20 0.31
GPR35 Q9HC97 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8727200 0.84 TRPV4 (0.38) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL7202604 0.84 TRPV4 (0.38) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL7768183 0.82 TRPV4 (0.36) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL8049906 0.82 TRPV4 (0.41) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL9489852 0.82 TRPV4 (0.42) TRPV4KHKCYP11B2CYP11B1EGLN2
SCHEMBL9447114 0.80 TRPV4 (0.35) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL30107963 0.79 TRPV4 (0.38) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL9693924 0.79 GPR35 (0.41) TRPV4KHKCYP11B2ALDH1A1AR
SCHEMBL7922013 0.79 TRPV4 (0.38) TRPV4KHKCYP11B2MAPK1ALDH1A1
SCHEMBL16122643 0.77 GRM5 (0.42) TRPV4KHKCYP11B2ALDH1A1VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635486-B1 Process for the preparation of fluorobenzonitriles CLARIANT GMBH (DE) 1998-12-09 EP disclosed
US-5777181-A 2, 4, 5-trihalogeno- and 2, 3, 4, 5-tetrahalogenobenzene derivatives BAYER AKTIENGESELLSCHAFT (DE) 1998-07-07 US disclosed
US-5565614-A FLUORINATION BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
US-5530158-A CHEMICAL INTERMEDIATE FOR ANTIBACTERIALS BAYER AKTIENGESELLSCHAFT (DE) 1996-06-25 US disclosed
US-5466859-A Process for preparing fluorobenzonitriles HOECHST AKTIENGESELLSCHAFT (DE) 1995-11-14 US disclosed
EP-0635486-A2 Process for the preparation of fluorobenzonitriles HOECHST AKTIENGESELLSCHAFT (DE) 1995-01-25 EP disclosed
US-5362909-A Two stage fluorination BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US disclosed
US-5200548-A Intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
US-5072038-A Chemical intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-10 US disclosed
CN-1013370-B Process for preparing derivatives of 2, 4, 5-trihalobenzenes and 2, 3, 4, 5-tetrahalobenzenes BAYER AG (DE) 1991-07-31 CN disclosed
EP-0164619-B1 2,4,5-TRIHALO OR 2,3,4,5-TETRAHALO BENZENE DERIVATIVES AND PROCESS FOR PRODUCING THEM BAYER AG (DE) 1988-10-12 EP disclosed
CN-85101737-A Preparation 2,4,5-trihalogenated benzene and 2,3,4, the derivative method of 5-tetrahalogeno-benzene 1987-01-31 CN disclosed
EP-0164619-A1 2,4,5-Trihalo or 2,3,4,5-tetrahalo benzene derivatives and process for producing them BAYER AG (DE) 1985-12-18 EP disclosed