SCHEMBL8664428

SCHEMBL8664428

O=C(Nc1c(Cl)cncc1Cl)c1cccc(OC(F)F)c1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 10/20 0.47
PDE4B Q07343 9/20 0.47
PDE4A P27815 3/20 0.47
PDE4C Q08493 2/20 0.47
ABCB11 O95342 1/20 0.47
SGMS2 Q8NHU3 4/20 0.45
P2RX7 Q99572 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29824898 1.00 PDE4D (0.47) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL7065703 0.83 PDE4A (0.54) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL23499796 0.80 PDE4B (0.69) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL7368887 0.80 PDE4B (0.64) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL29682915 0.80 PDE4B (0.69) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL2518447 0.77 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL8890462 0.73 PDE4B (0.71) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL6571717 0.72 PDE4D (0.61) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL5794099 0.71 PDE4D (0.65) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL14705239 0.71 PDE4B (0.65) PDE4DPDE4BPDE4APDE4CABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240316015-A1 COMPOSITION AND METHOD FOR TREATING TUMORS NATURAL MEDICINE INSTITUTE OF ZHEJIANG YANGSHENGTANG CO., LTD. (CN) 2024-09-26 US disclosed
EP-4282413-A1 COMPOSITION AND METHOD FOR TREATING TUMORS NATURAL MEDICINE INSTITUTE OF ZHEJIANG YANGSHENGTANG CO., LTD. (CN) 2023-11-29 EP disclosed
CN-116963773-A Compositions and methods for treating tumors 浙江养生堂天然药物研究所有限公司 2023-10-27 CN disclosed
CN-115397411-A Pharmaceutical combination and use thereof 浙江养生堂天然药物研究所有限公司 2022-11-25 CN disclosed
US-5712298-A Fluoroalkoxy-substituted benzamides and their use as cyclic nucleotide phosphodiesterase inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240316015-A1 COMPOSITION AND METHOD FOR TREATING TUMORS PDE4B, PDE4A, PDE4C PDE4D 4/4885PDE4B 1/4885PDE4A 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.