SCHEMBL8664720

SCHEMBL8664720

Cc1ccc(Cl)cc1N1C(=O)CN(C(C)C)C1=S

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 9/20 0.52
KMT2A Q03164 9/20 0.52
TSHR P16473 1/20 0.42
ALDH1A1 P00352 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
P2RX7 Q99572 1/20 0.37
HTR7 P34969 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
USP2 O75604 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661948 0.82 MEN1 (0.55) MEN1KMT2AALDH1A1NPSR1P2RX7
SCHEMBL8716448 0.78 KMT2A (0.64) MEN1KMT2AALDH1A1GAA
SCHEMBL8711085 0.77 KMT2A (0.51) MEN1KMT2AP2RX7GAA
SCHEMBL8915515 0.74 KMT2A (0.59) MEN1KMT2AALDH1A1GAA
SCHEMBL8663215 0.74 KMT2A (0.59) MEN1KMT2AALDH1A1GAA
SCHEMBL8711149 0.74 KMT2A (0.59) MEN1KMT2AALDH1A1NPSR1GAA
SCHEMBL7159612 0.73 MEN1 (0.47) MEN1KMT2ATSHRALDH1A1NPSR1
SCHEMBL8661222 0.73 MEN1 (0.48) MEN1KMT2AALDH1A1NPSR1P2RX7
SCHEMBL8479295 0.73 MEN1 (0.55) MEN1KMT2AALDH1A1P2RX7HTR7
SCHEMBL7655761 0.71 ALDH1A1 (0.42) MEN1KMT2ATSHRALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876355-A1 2-THIOXO-IMIDAZOLIDIN-4-ONE DERIVATIVES AND THEIR USE FOR INCREASING HDL CHOLESTEROL CONCENTRATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-11-11 EP claimed
US-5821372-A USEFUL FOR INCREASING BLOOD SERUM HIGH DENSITY LIPOPROTEIN LEVELS(HDL) AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-13 US claimed
WO-1997019932-A1 2-THIOXO-IMIDAZOLIDIN-4-ONE DERIVATIVES AND THEIR USE FOR INCREASING HDL CHOLESTEROL CONCENTRATION AMERICAN HOME PRODUCTS CORPORATION (US) 1997-06-05 WO claimed
US-5554607-A INCREASING HDL CHOLESTEROL AMERICAN HOME PRODUCTS CORPORATION (US) 1996-09-10 US claimed
US-5821372-A USEFUL FOR INCREASING BLOOD SERUM HIGH DENSITY LIPOPROTEIN LEVELS(HDL) AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-13 US disclosed
US-5554607-A INCREASING HDL CHOLESTEROL AMERICAN HOME PRODUCTS CORPORATION (US) 1996-09-10 US disclosed