SCHEMBL8668084

SCHEMBL8668084

CCC(CC)Nc1c(C(N)c2ccc(C#N)cc2)c(=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
CYP2A6 P11509 1/20 0.33
CYP19A1 P11511 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HTT P42858 1/20 0.32
ELANE P08246 1/20 0.32
CXCR2 P25025 2/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
F2R P25116 1/20 0.32
CXCR1 P25024 1/20 0.32
LSS P48449 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664139 0.82 ABCC9 (0.37) GRIA1GRIA2GRIA3GRIA4ABCC9
SCHEMBL8667527 0.80 ABCC9 (0.51) GRIA1GRIA2GRIA3GRIA4ABCC9
SCHEMBL8665101 0.75 ABCC9 (0.37) GRIA1GRIA2GRIA3GRIA4ABCC9
SCHEMBL7887143 0.75 LOXL2 (0.47) ABCC9ABCC8KCNJ11KCNJ8CYP2A6
SCHEMBL8666923 0.73 CYP19A1 (0.32) GRIA1GRIA2GRIA3GRIA4ABCC9
SCHEMBL15157661 0.67 SLC6A4 (0.52) GRIA1GRIA2GRIA3GRIA4CYP2A6
SCHEMBL8373592 0.64 ABCC9 (0.51) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL24181391 0.63 CYP2A6 (0.44) GRIA1GRIA2GRIA3GRIA4CYP2A6
SCHEMBL21562627 0.63 CYP2A6 (0.44) GRIA1GRIA2GRIA3GRIA4CYP2A6
SCHEMBL7894157 0.63 CXCR2 (0.39) ABCC9ABCC8KCNJ11KCNJ8CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846999-A Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 1998-12-08 US claimed
US-5846999-A Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 1998-12-08 US disclosed