SCHEMBL8669489

SCHEMBL8669489

COc1ccc(CCN2CCC(C=O)CC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.67
HRH3 Q9Y5N1 3/20 0.63
KCNJ1 P48048 1/20 0.56
KCNH2 Q12809 1/20 0.56
HTR1A P08908 1/20 0.54
SLC6A4 P31645 1/20 0.54
OPRM1 P35372 1/20 0.53
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493570 0.85 SIGMAR1 (0.58) SIGMAR1OPRM1
SCHEMBL12023880 0.82 SIGMAR1 (0.75) SIGMAR1HRH3HTR1ASLC6A4
SCHEMBL19609684 0.81 HRH1 (0.53) KCNJ1KCNH2OPRM1
SCHEMBL4069868 0.81 HTR2A (0.59) KCNJ1KCNH2
SCHEMBL10499190 0.81 SIGMAR1 (0.73) SIGMAR1HRH3KCNJ1KCNH2HTR1A
SCHEMBL7829844 0.80 ACHE (0.63) SIGMAR1KCNH2
SCHEMBL3590279 0.80 SIGMAR1 (0.58) SIGMAR1HRH3KCNJ1KCNH2HTR1A
Hydrochloric Acid SCHEMBL8502542 0.79 HTR2A (0.58) KCNJ1KCNH2
SCHEMBL7841889 0.79 SIGMAR1 (0.65) SIGMAR1HRH3KCNJ1KCNH2HTR1A
SCHEMBL3590284 0.79 SIGMAR1 (0.60) SIGMAR1HRH3KCNJ1KCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739150-A Piperidinyl thiacyclic derivatives MERRELL PHARMACEUTICALS INC. (US) 1998-04-14 US disclosed
EP-0626968-A4 1995-01-04 EP disclosed
EP-0626968-A1 PIPERIDINYL THIACYCLIC DERIVATIVES MERRELL PHARMACEUTICALS INC. (US) 1994-12-07 EP disclosed