SCHEMBL8669706

SCHEMBL8669706

NC(=O)c1c(C(=O)O)cccc1-c1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 2/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
SLC6A3 Q01959 1/20 0.51
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
SOS1 Q07889 1/20 0.49
HIF1A Q16665 1/20 0.49
MCL1 Q07820 1/20 0.47
FABP3 P05413 1/20 0.46
FABP4 P15090 1/20 0.46
FABP5 Q01469 1/20 0.46
HDAC4 P56524 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
GSTP1 P09211 1/20 0.45
FTO Q9C0B1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883731 0.89 ACMSD (0.55) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL28442421 0.86 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3HDAC4HDAC2
SCHEMBL84188 0.82 SLC6A2 (0.66) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL29916354 0.82 BCAT2 (0.63) FABP3FABP4FABP5ALDH1A1GAA
SCHEMBL30610922 0.82 SLC6A2 (0.66) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL570758 0.82 BCAT2 (0.63) FABP3FABP4FABP5ALDH1A1GAA
SCHEMBL29618929 0.82 SLC6A2 (0.66) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL31621280 0.81 SLC6A2 (0.64) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
Bromide SCHEMBL7032662 0.81 SLC6A2 (0.64) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL31621279 0.81 SLC6A2 (0.64) ACMSDSLC6A2SLC6A4SLC6A3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020138011-A1 TEREPHTHALIC ACID DERIVATIVE HAVING RING-FUSED STRUCTURE 第一三共株式会社 2020-07-02 WO disclosed
EP-0876330-A1 ARYL OR HETEROARYL AMIDES OF TETRAHYDRONAPHTHALENE, CHROMAN, THIOCHROMAN AND 1,2,3,4-TETRAHYDROQUINOLINE CARBOXYLIC ACIDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1998-11-11 EP disclosed
WO-1997019052-A1 ARYL OR HETEROARYL AMIDES OF TETRAHYDRONAPHTHALENE, CHROMAN, THIOCHROMAN AND 1,2,3,4-TETRAHYDROQUINOLINE CARBOXYLIC ACIDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1997-05-29 WO disclosed